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SMER3

●Purchase●DescriptionSmallMoleculeEnhancerofRapamycin3(SMER3)isaspecificinhibitoroftheubiquitinE3ligaseSCFMET30

  • 產品型號:27718-2
  • 廠商性質:生產廠家
  • 更新時間:2023-12-19
  • 訪  問  量:125
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Description

Small Molecule Enhancer of Rapamycin 3 (SMER3) is a specific inhibitor of the ubiquitin E3 ligase SCFMET30. SMER3 binds directly to the F-box subunit Met30 and blocks binding to the SCF core complex. Cell permeable. Significant inhibition is typically seen at 30-100 μM.

Synonyms
9H–Indeno[1,2–e][1,2,5]oxadiazolo[3,4–b]pyrazin–9–one
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